Molecule Details
InChIKeyOEFUMBDQRIIGBZ-UHFFFAOYSA-N
Compound Name6-tert-butylsulfonyl-7-methoxy-N-(2-methylphenyl)imidazo[1,2-a]pyridine-3-carboxamide
Canonical SMILESCOc1cc2ncc(C(=O)Nc3ccccc3C)n2cc1S(=O)(=O)C(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43353 RIPK2 Homo sapiens Human PF00619 PF07714 7.6 IC50 ChEMBL;BindingDB
P07948 LYN Homo sapiens Human PF07714 PF00017 PF00018 7.3 IC50 ChEMBL;BindingDB
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 6.9 IC50 ChEMBL;BindingDB