Molecule Details
InChIKeyOEAQKLHDOJQQKF-UHFFFAOYSA-N
Compound Name2-{3-Carboxy-2-[3-(4-sulfamoyl-phenyl)-thioureido]-propionylamino}-succinic acid
Canonical SMILESNS(=O)(=O)c1ccc(N/C(S)=N/C(CC(=O)O)C(=O)NC(CC(=O)O)C(=O)O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.65
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.8 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.8 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.3 Ki ChEMBL;BindingDB