Molecule Details
InChIKeyODTQXVXYPYSPSO-UHFFFAOYSA-N
Compound Name5-[3-[5-[(3,5-dichloro-4-pyridinyl)carbamoylamino]-1-ethyl-6-oxopyridazin-3-yl]phenyl]-3-N-[3-(dimethylamino)propyl]-1-N-ethylbenzene-1,3-dicarboxamide
Canonical SMILESCCNC(=O)c1cc(C(=O)NCCCN(C)C)cc(-c2cccc(-c3cc(NC(=O)Nc4c(Cl)cncc4Cl)c(=O)n(CC)n3)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 10.3 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 6.4 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB