Molecule Details
InChIKeyODNIEBFFNONVCK-UHFFFAOYSA-N
Compound Name5-[2-[4-(1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-3-methyl-6,7-dihydro-2H-pyrazolo[4,3-c]pyridin-4-one
Canonical SMILESCc1n[nH]c2c1C(=O)N(CCN1CCC(c3noc4ccccc34)CC1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB