Molecule Details
InChIKeyODJIGTDOQQQJKM-JKRBJUMTSA-N
Compound Name1-[[(2S,6R)-3-oxa-13-thiatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methyl]-4-phenylpiperidine
Canonical SMILESc1ccc(C2CCN(CC3C[C@@H]4c5ccccc5Sc5ccccc5[C@H]4O3)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35367 HRH1 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB