Molecule Details
InChIKeyOCZDPFMSAKKNRH-OQLLNIDSSA-N
Compound Name3-[[(E)-4-(dimethylamino)but-2-enoyl]amino]-N-[4-[[4-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)pyrimidin-2-yl]amino]phenyl]benzamide
Canonical SMILESCN(C)C/C=C/C(=O)Nc1cccc(C(=O)Nc2ccc(Nc3nccc(-c4c(-c5ccccc5)nn5ccccc45)n3)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 8.9 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB