Molecule Details
InChIKeyOCUYCOQPRGFQEV-UHFFFAOYSA-N
Compound Name2-fluoro-4-(4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)pyrimidin-2-ylamino)-N-methylbenzamide
Canonical SMILESCNC(=O)c1ccc(Nc2nccc(-c3cnc(C)n3C(C)C)n2)cc1F
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.41
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 9.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 9.0 pIC50 TTD_MultiTarget
Q00532 CDKL1 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB