Molecule Details
InChIKeyOCOGBPYFWRDLHI-RELWKKBWSA-N
Compound Name(E)-3-(4-hydroxy-3-methoxyphenyl)-N-[2-[2-(5-methoxy-1H-indol-3-yl)ethylamino]-2-oxoethyl]-N-[8-(1,2,3,4-tetrahydroacridin-9-ylamino)octyl]prop-2-enamide
Canonical SMILESCOc1ccc2[nH]cc(CCNC(=O)CN(CCCCCCCCNc3c4c(nc5ccccc35)CCCC4)C(=O)/C=C/c3ccc(O)c(OC)c3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06276 BCHE Homo sapiens Human PF08674 PF00135 7.6 IC50 ChEMBL;BindingDB
P22303 ACHE Homo sapiens Human PF08674 PF00135 7.4 IC50 ChEMBL;BindingDB