Molecule Details
InChIKeyOCHMDWMGQAQDSI-HGYOODBQSA-N
Compound NameH-2Fpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-2Fpa-NH2
Canonical SMILESCC(C)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccnc2)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc2ccccc2F)CSSC[C@H](C(=O)N[C@@H](Cc2ccccc2F)C(N)=O)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30872 SSTR1 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P30874 SSTR2 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB