Molecule Details
InChIKeyOBZHEBDUNPOCJG-WBXJDKIVSA-N
Compound NameCarbenoxolone
Canonical SMILESCC1(C)[C@@H](OC(=O)CCC(=O)O)CC[C@]2(C)[C@H]3C(=O)C=C4[C@@H]5C[C@@](C)(C(=O)O)CC[C@]5(C)CC[C@@]4(C)[C@]3(C)CC[C@@H]12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB02329
Drug NameCarbenoxolone
CAS Number5697-56-3
Groups experimental
ATC Codes A02BX01 A02BX71 A02BX51
DescriptionAn agent derived from licorice root. It is used for the treatment of digestive tract ulcers, especially in the stomach. Antidiuretic side effects are frequent, but otherwise the drug is low in toxicity. [PubChem]

Categories: Alimentary Tract and Metabolism Anti-Ulcer Agents Drugs for Acid Related Disorders Drugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord) Gastrointestinal Agents Pentacyclic Triterpenes Terpenes Triterpenes
Cross-references: BindingDB: 50247012 CHEMBL499915 ChemSpider: 552190 PDB: CBO PubChem:636403 PubChem:46508820 RxCUI: 2017 Therapeutic Targets Database: DNC000388 Wikipedia: Carbenoxolone ZINC: ZINC000003977823
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P80365 HSD11B2 Homo sapiens Human PF00106 6.8 IC50 ChEMBL;BindingDB
P28845 HSD11B1 Homo sapiens Human PF00106 6.5 IC50 ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P19992 P19992 3-alpha-(or 20-beta)-hydroxysteroid dehydrogenase binder targets
P28845 HSD11B1 11-beta-hydroxysteroid dehydrogenase 1 inhibitor targets