Molecule Details
InChIKeyOAWZSUHVKPQVIU-LEEDBYTESA-N
Canonical SMILESCOc1ccc([C@H](Cc2c(Cl)c[n+]([O-])cc2Cl)OC(=O)c2ccc(CN[C@@H](C(=O)O[C@H]3CN4CCC3CC4)c3ccccc3)s2)cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.5
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P20309 CHRM3 Homo sapiens Human PF00001 10.2 Ki ChEMBL
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 8.8 IC50 ChEMBL