Molecule Details
InChIKeyOAUFPDQMACFAMN-UHFFFAOYSA-N
Compound Name3-[2-[4-(2-chlorophenyl)-1-piperazinyl]ethyl]-6-(4-methylphenyl)-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione
Canonical SMILESCc1ccc(-c2cc3c(=O)n(CCN4CCN(c5ccccc5Cl)CC4)c(=O)[nH]c3[nH]2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P25100 ADRA1D Homo sapiens Human PF00001 7.9 Ki ChEMBL
P35348 ADRA1A Homo sapiens Human PF00001 7.9 Ki ChEMBL
P35368 ADRA1B Homo sapiens Human PF00001 7.9 Ki ChEMBL
P21728 DRD1 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB