Molecule Details
InChIKeyOAIDOYYRSBXKJG-CMDGGOBGSA-N
Compound NameN-[3-[(E)-2-[5-(methanesulfonamido)-6-pyrrolidin-1-yl-1H-indazol-3-yl]ethenyl]phenyl]-4-methylpiperazine-1-carboxamide
Canonical SMILESCN1CCN(C(=O)Nc2cccc(/C=C/c3n[nH]c4cc(N5CCCC5)c(NS(C)(=O)=O)cc34)c2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.97
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget