Molecule Details
InChIKeyOAEWNSKRLBVVBV-OBTVHEKISA-N
Compound Name(2R,3S,4R)-1-[2-(dibutylamino)-2-oxoethyl]-2-(2,2-dimethylpentyl)-4-(7-methoxy-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
Canonical SMILESCCCCN(CCCC)C(=O)CN1C[C@@H](c2cc(OC)c3c(c2)OCO3)[C@H](C(=O)O)[C@H]1CC(C)(C)CCC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.17
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.3 Ki ChEMBL
P08908 HTR1A Homo sapiens Human PF00001 6.7 Ki ChEMBL
Q99720 SIGMAR1 Homo sapiens Human PF04622 6.5 Ki ChEMBL