Molecule Details
InChIKeyNZTHPWQOSONJAR-UHFFFAOYSA-N
Compound Name6-Chloro-4-methyl-11-[2-(4-phenylpiperazin-1-yl)ethylamino]-4,5,9,10-tetrazatricyclo[7.4.0.02,7]trideca-1,5,7,10,12-pentaen-3-one
Canonical SMILESCn1nc(Cl)c2cn3nc(NCCN4CCN(c5ccccc5)CC4)ccc3c2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB