Molecule Details
InChIKeyNZQDWKCNBOELAI-KSFYIVLOSA-N
Canonical SMILESO=C(O)c1ccc(C(F)(F)F)cc1-c1ccc2c(c1)OC[C@H](Cc1ccccc1)[C@H]2O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB13053
Drug NameCP-195543
CAS Number204981-48-6
Groups investigational
ATC Codes nan
DescriptionCP-195,543 has been used in trials studying the treatment of Arthritis, Rheumatoid.

Categories: Benzopyrans Heterocyclic Compounds, Fused-Ring Pyrans
Cross-references: BindingDB: 50215854 CHEMBL301829 ChemSpider: 7999633 PubChem:9823886 PubChem:347829182
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15722 LTB4R Homo sapiens Human PF00001 8.0 IC50 ChEMBL
Q9NPC1 LTB4R2 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
DrugBank Target Actions (1)
Target Gene Target Name Action Type
Q15722 LTB4R Leukotriene B4 receptor 1 antagonist targets