Molecule Details
InChIKeyNZGWRTVGHIZQDX-UHFFFAOYSA-N
Compound Name7,8-dimethoxy-2-[4-(4-pyridin-2-ylpiperazin-1-yl)butyl]-4,5-dihydro-3H-2-benzazepin-1-one
Canonical SMILESCOc1cc2c(cc1OC)C(=O)N(CCCCN1CCN(c3ccccn3)CC1)CCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB