Molecule Details
InChIKeyNYVUSSXLPQHLMH-UHFFFAOYSA-N
Compound Name2-Amino-N-[4-Methoxy-3-(Trifluoromethyl)phenyl]-4-Methyl-3-[2-(Methylamino)quinazolin-6-Yl]benzamide
Canonical SMILESCNc1ncc2cc(-c3c(C)ccc(C(=O)Nc4ccc(OC)c(C(F)(F)F)c4)c3N)ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 8.0 IC50 ChEMBL;BindingDB
Q9NZJ5 EIF2AK3 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
Q9P2K8 EIF2AK4 Homo sapiens Human PF12745 PF00069 PF05773 PF13393 6.4 IC50 ChEMBL;BindingDB