Molecule Details
InChIKeyNYHVIVWBHLTODF-UHFFFAOYSA-N
Compound NameN-(Phenyl)-1H-pyrazol-4-yl]-1-(phenylsulfonyl)-1H-pyrrolo-[2,3-b]pyridin-2-yl]phenyl}acetamide
Canonical SMILESCCn1cc(-c2ccnc3[nH]c(-c4ccc(NC(C)=O)cc4)cc23)c(-c2ccc(NC(=O)Nc3ccccc3)cc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget