Molecule Details
InChIKeyNYGHGTMKALXFIA-UHFFFAOYSA-N
Compound NameAzapetine
Canonical SMILESC=CCN1Cc2ccccc2-c2ccccc2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB13727
Drug NameAzapetine
CAS Number146-36-1
Groups experimental
ATC Codes C04AX30
Descriptionnan

Categories: Heterocyclic Compounds, Fused-Ring Peripheral Vasodilators
Cross-references: BindingDB: 81805 ChEBI: 134955 CHEMBL2110596 ChemSpider: 8620 Wikipedia: Azapetine ZINC: ZINC000001481977
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 7.4 Ki BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.0 Kd ChEMBL
P35348 ADRA1A Homo sapiens Human PF00001 7.0 Kd ChEMBL
P35368 ADRA1B Homo sapiens Human PF00001 7.0 Kd ChEMBL