Molecule Details
InChIKeyNXZVLIWBXMLTSL-UHFFFAOYSA-N
Compound Name8-anilino-N-(2-hydroxyethyl)-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Canonical SMILESCn1nc(C(=O)NCCO)c2c1-c1nc(Nc3ccccc3)ncc1CC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.1 pIC50 TTD_MultiTarget
O14965 AURKA Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB