Molecule Details
InChIKeyNXXSVEQIIURRGX-UHFFFAOYSA-N
Compound Name4-[7-(3-aminopropoxy)-1-ethyl-4-(1H-pyrrol-2-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine
Canonical SMILESCCn1c(-c2nonc2N)nc2c(-c3ccc[nH]3)ncc(OCCCN)c21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15418 RPS6KA1 Homo sapiens Human PF00069 PF00433 7.9 IC50 ChEMBL;BindingDB
P31749 AKT1 Homo sapiens Human PF00169 PF00069 PF00433 7.5 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 6.8 IC50 ChEMBL;BindingDB