Molecule Details
InChIKeyNXWZJBVSPZNPCA-UHFFFAOYSA-N
Compound NameN-benzyl-N-[6-cyano-1-[(3-methylimidazol-4-yl)methyl]-3,4-dihydro-2H-quinolin-3-yl]-1-methylpyrazole-4-sulfonamide
Canonical SMILESCn1cc(S(=O)(=O)N(Cc2ccccc2)C2Cc3cc(C#N)ccc3N(Cc3cncn3C)C2)cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.34
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.3 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.3 IC50 ChEMBL