Molecule Details
InChIKeyNXTMDUWTQZXRRK-GXCCDKSUSA-N
Compound Namecyclo[Asu(NHOH)(NHOH)-D-Tyr(Me)-Ile-D-Pro]
Canonical SMILESCC[C@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13547 HDAC1 Homo sapiens Human PF00850 9.4 IC50 ChEMBL;BindingDB
P56524 HDAC4 Homo sapiens Human PF12203 PF00850 8.5 IC50 ChEMBL;BindingDB