Molecule Details
InChIKeyNXJYLDGTQWINTD-UHFFFAOYSA-N
Compound NameN-[6-[(4-amino-6,7-dimethoxyquinazolin-2-yl)-methylamino]hexyl]-N-methyl-2,3-dihydro-1,4-benzodioxine-3-carboxamide
Canonical SMILESCOc1cc2nc(N(C)CCCCCCN(C)C(=O)C3COc4ccccc4O3)nc(N)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35368 ADRA1B Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB