Molecule Details
InChIKeyNWCLUPOGVWVFRT-OLILMLBXSA-N
Compound Name(3S)-N-[2-(1H-benzimidazol-2-ylmethylamino)-2-oxoethyl]-2-[(2R)-3-(4-hydroxy-2,6-dimethylphenyl)-2-methylpropyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Canonical SMILESCc1cc(O)cc(C)c1C[C@@H](C)CN1Cc2ccccc2C[C@H]1C(=O)NCC(=O)NCc1nc2ccccc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41143 OPRD1 Homo sapiens Human PF00001 10.5 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB