Molecule Details
InChIKeyNVMGBEWNMCNKHG-HNNXBMFYSA-N
Canonical SMILESCNC(=O)C[C@H]1COc2cc(F)c(CC(C)C)cc2N1C(=O)c1ccnc(NC(N)=O)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08235 NR3C2 Homo sapiens Human PF00104 PF00105 7.5 IC50 ChEMBL;BindingDB
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 6.9 Ki ChEMBL;BindingDB