Molecule Details
InChIKeyNVIMRDPIWGJULC-CYBMUJFWSA-N
Compound Name(R)-1-(6-(5-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazolo[3,4-c]pyridin-3-yl)pyridin-2-yl)pyrrolidin-3-amine
Canonical SMILESCn1cc(-c2cc3c(-c4cccc(N5CC[C@@H](N)C5)n4)n[nH]c3cn2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.8 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.9 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB