Molecule Details
InChIKeyNUQNGPSYNHDQBA-UHFFFAOYSA-N
Compound Name6-(6-Phenylmethoxypyrazin-2-yl)-1-(6-piperazin-1-yl-2-pyridinyl)pyrazolo[4,3-c]pyridine
Canonical SMILESc1ccc(COc2cncc(-c3cc4c(cn3)cnn4-c3cccc(N4CCNCC4)n3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.5 Ki ChEMBL;BindingDB