Molecule Details
InChIKeyNUBKAVGOKIBUDW-DZDBGDIESA-N
Compound NameH-2Nal-Cys(1)-3Pal-D-Trp-Lys-D-Val-D-Cys(1)-Dip-NH2
Canonical SMILESCC(C)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccnc2)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc2ccc3ccccc3c2)CSSC[C@H](C(=O)N[C@H](C(N)=O)C(c2ccccc2)c2ccccc2)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30874 SSTR2 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P35346 SSTR5 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB