Molecule Details
InChIKeyNTYJRAGMLUHRNV-DZGOFYRVSA-N
Compound NameH-Tyr-D-Ala-Gly-Phe-Pro-Trp-Unk
Canonical SMILESC[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25103 TACR1 Homo sapiens Human PF00001 10.0 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.2 Ki ChEMBL