Molecule Details
InChIKeyNTSDIJMNXYJJNG-SFHVURJKSA-N
Compound NameAzd-5597
Canonical SMILESCN[C@H]1CCN(C(=O)c2ccc(Nc3ncc(F)c(-c4cnc(C)n4C(C)C)n3)cc2)C1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.7
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 8.7 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 8.7 pIC50 TTD_MultiTarget