Molecule Details
InChIKeyNTCOZURJKJMLEZ-UHFFFAOYSA-N
Compound Name4-(dimethylamino)-N-[3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-2,4-dioxo-1H-[1]benzothiolo[3,2-d]pyrimidin-8-yl]butanamide
Canonical SMILESCOc1ccccc1N1CCN(CCn2c(=O)[nH]c3c(sc4ccc(NC(=O)CCCN(C)C)cc43)c2=O)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25100 ADRA1D Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB