Molecule Details
InChIKeyNTBBSTMZDUINTQ-UHFFFAOYSA-N
Compound Name6-[[1-[1-(2-methylquinolin-5-yl)oxypropan-2-yl]piperidin-4-yl]methyl]-4H-1,4-benzoxazin-3-one
Canonical SMILESCc1ccc2c(OCC(C)N3CCC(Cc4ccc5c(c4)NC(=O)CO5)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB