Molecule Details
InChIKeyNSQXHPWPAPWSLN-UHFFFAOYSA-N
Compound NameN-{4-[4-(2-{3-[(dimethylamino)methyl]phenyl}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1-ethyl-1H-pyrazol-3-yl]phenyl}-N'-ethylurea
Canonical SMILESCCNC(=O)Nc1ccc(-c2nn(CC)cc2-c2ccnc3[nH]c(-c4cccc(CN(C)C)c4)cc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.9 pIC50 TTD_MultiTarget