Molecule Details
InChIKeyNSNKKSURBOMEKE-UHFFFAOYSA-N
Compound NameN-[5-[6-(4-methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]acetamide
Canonical SMILESCOc1cc(C)c(-c2cc(-c3cnc(NC(C)=O)s3)nc(-c3cnccn3)n2)c(C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53671 LIMK2 Homo sapiens Human PF00412 PF00595 PF07714 7.2 IC50 ChEMBL;BindingDB
P53667 LIMK1 Homo sapiens Human PF00412 PF00595 PF07714 7.1 IC50 ChEMBL;BindingDB
Q96S53 TESK2 Homo sapiens Human PF07714 6.2 IC50 ChEMBL;BindingDB