Molecule Details
InChIKeyNRTIHDQHAKWSTG-UHFFFAOYSA-N
Compound Name4-(3,4-Dichlorophenyl)-7-(pyridazin-3-yl)-1,2,3,4-tetrahydroisoquinoline
Canonical SMILESClc1ccc(C2CNCc3cc(-c4cccnn4)ccc32)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.2 IC50 ChEMBL;BindingDB
Q01959 SLC6A3 Homo sapiens Human PF00209 7.8 IC50 ChEMBL;BindingDB
P23975 SLC6A2 Homo sapiens Human PF00209 7.6 IC50 ChEMBL;BindingDB