Molecule Details
InChIKeyNRSNOIKPAFOCRX-UHFFFAOYSA-N
Compound Name1-(3-Methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[5,4-d]pyrimidine
Canonical SMILESCOc1cccc(-n2ncc3c(N4CCN(c5ccccc5OC)CC4)ncnc32)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11169 SLC2A3 Homo sapiens Human PF00083 6.8 IC50 ChEMBL;BindingDB
P11166 SLC2A1 Homo sapiens Human PF00083 6.7 IC50 ChEMBL;BindingDB
P11168 SLC2A2 Homo sapiens Human PF00083 6.0 IC50 ChEMBL;BindingDB