Molecule Details
InChIKeyNRHCLLDEPJFJNY-UHFFFAOYSA-N
Compound Name4-(bis(4-methylpiperidin-1-yl)amino)-N-(4-sulfamoylphenyl)butanamide
Canonical SMILESCC1CCN(N(CCCC(=O)Nc2ccc(S(N)(=O)=O)cc2)N2CCC(C)CC2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.74
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 7.0 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.6 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.6 pIC50 TTD_MultiTarget