Molecule Details
InChIKeyNRGHCWQGTHPFTE-FVWCLLPLSA-N
Compound Name(4aR,5aS,8aR,13aS,15aS,15bR)-10-amino-4a,5,5a,7,8,13a,15,15a,15b,16-decahydro-2H-4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one
Canonical SMILESNc1ccc2c(c1)[C@@]13CCN4CC5=CCO[C@H]6CC(=O)N2[C@H]1[C@H]6[C@H]5C[C@H]43
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P23415 GLRA1 Homo sapiens Human PF02931 PF02932 7.1 IC50 ChEMBL;BindingDB
P48167 GLRB Homo sapiens Human PF02931 PF02932 6.6 IC50 ChEMBL