Molecule Details
InChIKeyNQZUDRUZBFMADH-UHFFFAOYSA-N
Compound NameN-[3-[3,3,6,6-tetramethyl-1,8-dioxo-10-(4-sulfamoylphenyl)-4,5,7,9-tetrahydro-2H-acridin-9-yl]phenyl]naphthalene-2-sulfonamide
Canonical SMILESCC1(C)CC(=O)C2=C(C1)N(c1ccc(S(N)(=O)=O)cc1)C1=C(C(=O)CC(C)(C)C1)C2c1cccc(NS(=O)(=O)c2ccc3ccccc3c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 6.3 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB
O43570 CA12 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB