Molecule Details
InChIKeyNQRKYASMKDDGHT-UHFFFAOYSA-N
Canonical SMILESNOCC(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.12
SourceChEMBL
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB02079
Drug NameAminooxyacetic acid
CAS Number645-88-5
Groups experimental
ATC Codes nan
DescriptionA compound that inhibits aminobutyrate aminotransferase activity in vivo, thereby raising the level of gamma-aminobutyric acid in tissues. [PubChem]

Categories: Acetates Acids, Acyclic Amines Enzyme Inhibitors GABA Agents Hydroxylamines Neurotransmitter Agents
Cross-references: ChEBI: 40823 CHEMBL347862 ChemSpider: 280 PDB: AOA PubChem:286 PubChem:46507597 Wikipedia: Aminooxyacetic_acid ZINC: ZINC000004689151
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32929 CTH Homo sapiens Human PF01053 6.2 IC50 ChEMBL
P35520 CBS Homo sapiens Human PF00571 PF00291 6.0 IC50 ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P21549 AGXT Alanine--glyoxylate aminotransferase binder targets
P35520 CBS Cystathionine beta-synthase inhibitor targets