Molecule Details
InChIKeyNQBOWNPIRYVPJI-UHFFFAOYSA-N
Canonical SMILESCCOc1ccc(-c2nc3ccccn3c2-c2ccnc(Nc3ccc(N4CCC(N5CCCCC5)CC4)c(C)c3OC)n2)cc1C(=O)Nc1c(F)cccc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06213 INSR Homo sapiens Human PF00757 PF17870 PF07714 PF01030 7.0 IC50 ChEMBL
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 7.0 IC50 ChEMBL