Molecule Details
InChIKeyNPATVCXCHCPFCB-OAHLLOKOSA-N
Compound Name(R)-2-(Benzylamino-methyl)-3,4,7,9-tetrahydro-2H-pyrano[2,3-e]indol-8-one
Canonical SMILESO=C1Cc2c(ccc3c2O[C@@H](CNCc2ccccc2)CC3)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB