Molecule Details
InChIKeyNNZRYGISYKGSCW-UHFFFAOYSA-N
Compound Name4-[3-(1H-benzimidazol-2-yloxy)phenyl]-7,7-dimethyl-4,6,8,9-tetrahydro-1H-pyrazolo[5,4-b]quinolin-5-one
Canonical SMILESCC1(C)CC(=O)C2=C(C1)Nc1n[nH]cc1C2c1cccc(Oc2nc3ccccc3[nH]2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
Q9NQS7 INCENP Homo sapiens Human PF03941 PF12178 8.1 IC50 ChEMBL
O14965 AURKA Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB