Molecule Details
InChIKeyNNDFRIHFDHSKHD-UHFFFAOYSA-N
Compound Name4-[[1-[3-[(4-Bromobenzoyl)amino]phenyl]-3-piperidin-1-ylpropyl]amino]quinazoline-8-carboxamide
Canonical SMILESNC(=O)c1cccc2c(NC(CCN3CCCCC3)c3cccc(NC(=O)c4ccc(Br)cc4)c3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.4 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 9.1 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.1 IC50 ChEMBL;BindingDB