Molecule Details
InChIKeyNNCWGHBKJIEMSS-UHFFFAOYSA-N
Compound Name8-[(4-Methoxypiperidin-4-yl)methoxy]-2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)quinoline
Canonical SMILESCOC1(COc2cccc3ccc(-c4nnc5ccccn45)nc23)CCNCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB