Molecule Details
InChIKeyNMULSNNATHYGPZ-UHFFFAOYSA-N
Compound NameN1-(4-(2-(4-(1H-benzo[d]imidazol-2-ylamino)naphthalen-1-yloxy)pyridin-3-yl)pyrimidin-2-yl)-N3,N3,2,2-tetramethylpropane-1,3-diamine
Canonical SMILESCN(C)CC(C)(C)CNc1nccc(-c2cccnc2Oc2ccc(Nc3nc4ccccc4[nH]3)c3ccccc23)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.44
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02763 TEK Homo sapiens Human PF00041 PF10430 PF07714 7.1 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.1 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.1 IC50 ChEMBL;BindingDB