Molecule Details
InChIKeyNMIXBOUDRDWICA-OOAXWGSJSA-N
Compound Namerac-5,7-difluoro-3-hydroxy-2,2-dimethyl-6-(3-methyl-1H-indol-7-yl)-2,3-dihydroquinolin-4(1H)-one O-ethyl oxime
Canonical SMILESCCO/N=C1/c2c(cc(F)c(-c3cccc4c(C)c[nH]c34)c2F)NC(C)(C)C1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 8.6 IC50 ChEMBL;BindingDB
P06401 PGR Homo sapiens Human PF00104 PF02161 PF00105 7.6 Ki ChEMBL;BindingDB
P10275 AR Homo sapiens Human PF02166 PF00104 PF00105 6.4 Ki ChEMBL;BindingDB