Molecule Details
InChIKeyNLZHOJOCWCLWFT-UHFFFAOYSA-N
Compound Name5-{4-[3-(2-Methylpyrimidin-5-yl)phenyl]piperazin-1-yl}pyrimidine-2,4-diamine
Canonical SMILESCc1ncc(-c2cccc(N3CCN(c4cnc(N)nc4N)CC3)c2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.1 IC50 ChEMBL;BindingDB
Q27783 Trypanosoma brucei brucei Pathogen PF00186 PF00303 8.7 IC50 BindingDB